ZM 241385

ZM 241385

CAT N°: 20447
Price:

From 48.00 40.80

ZM 241385 is a potent antagonist of A2A adenosine receptors (pIC50 = 9.52 for displacement of 5’-N-ethylcarboxamidoadenosine from rat phaeochromocytoma cell membranes).{32870,27926} It displays little or no activity at other A adenosine receptors. ZM 241385 is active in vivo.{32869,32871} It acts as an inverse agonist at constitutively active mutants of the human A2B adenosine receptor.{32641}

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