SCH 202676 (hydrobromide)

Biochemicals - Receptor Pharmacology

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Cat No: 16945

Biochemicals - Receptor Pharmacology

SCH 202676 is a reversible inhibitor of both agonist and antagonist binding to diverse G protein-coupled receptors (GPCRs).{27649} It blocks the binding of radiolabeled ligands to human opioid, adrenergic, muscarinic, dopaminergic, adenosine, and puri...

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Territorial Availability: Available through Bertin Technologies only in France

Synonyms:

N-(2,3-diphenyl-1,2,4-thiadiazol-5(2H)-ylidene)-methanamine, monohydrobromide

Correlated keywords:

70375-43-8 311814-53-6, 1056712-53-8 biochemicals inhibitors receptor biochemistry neuroscience SCH202676 HBr hydrobromic acid modulator GPCR G protein-coupled reversible inhibit agonist antagonist binding thiol modification

Product Overview:
SCH 202676 is a reversible inhibitor of both agonist and antagonist binding to diverse G protein-coupled receptors (GPCRs).{27649} It blocks the binding of radiolabeled ligands to human opioid, adrenergic, muscarinic, dopaminergic, adenosine, and purinergic receptors.{27649,27648,27647} It displays IC50 values of 0.1 to 1.8 µM for modulating ligand binding.{27649,27648} SCH 202676 may modulate GPCRs via thiol modification.{27646}

Size	5 mg
Shipping	dry ice
CAS Number	265980-25-4
Molecular Formula	C₁₅H₁₃N₃S • HBr
SMILES	C/N=C1SN(C2=CC=CC=C2)C(C3=CC=CC=C3)=N\1.Br
Molecular Weight	348,3
Formulation	A crystalline solid
Purity	≥95%
Custom Code	2930.90
UNSPSC code	12352100

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MSDS

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Our scientists are experts in the synthesis, purification, and characterization of biochemicals ranging from small drug-like heterocycles to complex biolipids, fatty acids, and many others. We are also highly skilled in all aspects of assay and antibody development, protein expression, crystallization, and structure determination.

Over the past thirty years, Cayman developed a deep knowledge base in lipid biochemistry, including research involving the arachidonic acid cascade, inositol phosphates, and cannabinoids. This knowledge enabled the production of reagents of exceptional quality for cancer, oxidative injury, epigenetics, neuroscience, inflammation, metabolism, and many additional lines of research.

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