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Oxybutynin (hydrochloride)

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    Oxybutynin (hydrochloride)
  • Oxybutynin (hydrochloride)
Cat No: 23825
Biochemicals - Receptor Pharmacology
Cayman

Oxybutynin is an antagonist of muscarinic acetylcholine receptors (Kis = 5, 14.5, 3.7, 5.3, and 40 nM for human recombinant M1-5, respectively).{39586} It inhibits intracellular calcium mobilization induced by carbamoylcholine (carbachol; Item No. 144...

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Territorial Availability: Available through Bertin Technologies only in France
Synonyms:
  • 4-(diethylamino)-2-butyn-1-yl ester ?-cyclohexyl-?-hydroxy-benzeneacetic acid, monohydrochloride
Correlated keywords:
  • 119579-36-1 1552323-10-0 5633-20-5 99937-06-1 Ditropan Lenditro Lyrinel XL chloride Cystrin Dridase Gelnique MJ43091 MJ-50-58 MJ50-58 MJ5058 Neoxy-Tape Pollakisu Tropax Benzeneacetic acid Cyclohexaneglycolic 43091 4309
Product Overview:
Oxybutynin is an antagonist of muscarinic acetylcholine receptors (Kis = 5, 14.5, 3.7, 5.3, and 40 nM for human recombinant M1-5, respectively).{39586} It inhibits intracellular calcium mobilization induced by carbamoylcholine (carbachol; Item No. 14486) in bladder smooth muscle and submandibular gland cells isolated from cynomolgus monkeys (Kis = 2 and 1 nM, respectively).{39587} Oxybutynin inhibits volume-induced bladder contraction (VIBC) and oxotremorine-induced salivation (OIS) in rats (ID50s = 0.062 and 0.089 mg/kg, respectively).{39586} It also increases pupil diameter (PD) and locomotor activity (LMA; ED50s = 0.29 and 0.52 mg/kg, respectively) and decreases small intestinal transit (SIT; ID50 = 0.22 mg/kg) in rats. Formulations containing oxybutynin have been used in the treatment of overactive bladder.
Size 1 g
Shipping dry ice
CAS Number 1508-65-2
Molecular Formula C22H31NO3 • HCl
SMILES OC(C1CCCCC1)(C(OCC#CCN(CC)CC)=O)C2=CC=CC=C2.Cl
Molecular Weight 394
Formulation A crystalline solid
Purity ≥98%
Custom Code 2914.50
UNSPSC code 12352100

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Our scientists are experts in the synthesis, purification, and characterization of biochemicals ranging from small drug-like heterocycles to complex biolipids, fatty acids, and many others. We are also highly skilled in all aspects of assay and antibody development, protein expression, crystallization, and structure determination.

Over the past thirty years, Cayman developed a deep knowledge base in lipid biochemistry, including research involving the arachidonic acid cascade, inositol phosphates, and cannabinoids. This knowledge enabled the production of reagents of exceptional quality for cancer, oxidative injury, epigenetics, neuroscience, inflammation, metabolism, and many additional lines of research.

Our organic and analytical chemists specialize in the rapid development of manufacturing processes and analytical methods to carry out clinical and commercial GMP-API production. Pre-clinical drug discovery efforts are currently underway in the areas of bone restoration and repair, muscular dystrophy, oncology, and inflammation. A separate group of Ph.D.-level scientists are dedicated to offering Hit-to-Lead Discovery and Profiling Services for epigenetic targets. Our knowledgeable chemists can be contracted to perform complete sample analysis for analytes measured by the majority of our assays. We also offer a wide range of analytical services using LC-MS/MS, HPLC, GC, and many other techniques.

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