Paynantheine (Item No. 21841) is an alkaloid of the herbal drug M. speciosa (also known as kratom). Kratom (mitragynine; Item Nos. 11151 | 18567) has opioid-like and stimulant effects, and paynantheine can be detected in urine after kratom ingestion.{20201} Paynantheine blocks the delayed-rectifier potassium current in human induced pluripotent stem cell-derived cardiomyocytes (IC50 = 2.47 µM), suggesting that it may have cardiotoxic effects.{33930} This product is intended for research and forensic applications.
Territorial Availability: Available through Bertin Technologies only in France
Technical Warning: Bertin Technologies restricts the sale of this product to licensed controlled substance laboratories and qualified academic research institutions. Please contact us for further details.
Special Advice: Please check regulation status before ordering; additionel fees can apply.
| Size | 1 mg, 5 mg, 500 µg |
|---|---|
| Shipping | dry ice |
| CAS number | 4697-66-9 |
| Molecular formula | C23H28N2O4 |
| Smiles | COC1=CC=CC2=C1C3=C([C@@](C[C@H](/C(C(OC)=O)=COC)[C@@H](C=C)C4)([H])N4CC3)N2, COC1=CC=CC2=C1C3=C([C@@](C[C@H](/C(C(OC)=O)=COC)[C@@H](C=C)C4)([H])N4CC3)N2, COC1=CC=CC2=C1C3=C([C@@](C[C@H](/C(C(OC)=O)=COC)[C@@H](C=C)C4)([H])N4CC3)N2 |
| Molecular weight | 396,5 |
| Custom code | 3822.19 |
| Formulation | A crystalline solid |
| Purity | ≥98% |
| UNSPSC code | 12352100 |
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