From €254.00 €215.90
8-iso-17-phenyl trinor Prostaglandin F2? (8-iso-17-phenyl trinor PGF2?) is the C-8 epimer of bimatoprost (free acid), a metabolically stable analog of PGF2?. Bimatoprost (free acid) binds to the FP receptor on ovine luteal cells with a relative potency of 756% compared to that of PGF2?.{2058} At the rat recombinant FP receptor expressed in CHO cells bimatoprost inhibits PGF2? binding with a Ki of 1.1 nM.{1374} There are no published studies of the pharmacological properties of 8-iso-17-phenyl trinor PGF2?.
Territorial Availability: Available through Bertin Technologies only in France
| Size | 1 mg, 10 mg, 5 mg |
|---|---|
| Shipping | dry ice |
| Molecular formula | C23H32O5 |
| Smiles | O[C@@H]1[C@@H](C/C=CCCCC(O)=O)[C@@H](/C=C/[C@@H](O)CCC2=CC=CC=C2)[C@H](O)C1, O[C@@H]1[C@@H](C/C=CCCCC(O)=O)[C@@H](/C=C/[C@@H](O)CCC2=CC=CC=C2)[C@H](O)C1, O[C@@H]1[C@@H](C/C=CCCCC(O)=O)[C@@H](/C=C/[C@@H](O)CCC2=CC=CC=C2)[C@H](O)C1 |
| Molecular weight | 388,5 |
| Custom code | 2937.50 |
| Formulation | A solution in methyl acetate |
| Purity | >98% |
| UNSPSC code | 12352100 |
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Our scientists are experts in the synthesis, purification, and characterization of biochemicals ranging from small drug-like heterocycles to complex biolipids, fatty acids, and many others. We are also highly skilled in all aspects of assay and antibody development, protein expression, crystallization, and structure determination.
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